5-HT1 | |
- Agonisti': 8-OH-DPAT
- Adatanserin
- Amfetamin
- Antidepresivi (npr. etoperidon, hidroksinefazodon, nefazodon, trazodon, triazoledion, vilazodon, vortioksetin)
- Atipični antipsihotici (npr. aripiprazol, asenapin, brekspiprazol, kariprazin, klozapin, lurasidon, kvetiapin, ziprasidon)
- Azapironi (npr. buspiron, eptapiron, gepiron, perospiron, tandospiron)
- Bay R 1531
- Befiradol
- BMY-14802
- Kanabidiol
- Dimemebfe
- Dopamin
- Ebalzotan
- Eltoprazin
- Enciprazin
- Enciprazin
- Ergolin (npr. bromokriptin, kabergolin, dihidroergotamin, ergotamin, lisurid, LSD, metilergometrin (metilergonovin), metisergid, pergolid)
- F-11461
- F-12826
- F-13714
- F-14679
- F-15063
- F-15599
- Flesinoxan
- Flibanserin
- Flumeksadol
- Hipidon
- Lesopitron
- LY-293284
- LY-301317
- mCPP
- MKC-242
- Naluzotan
- NBUMP
- Osemozotan
- Oksaflozan
- Pardoprunoks
- Piklozotan
- Rauwolscin
- Repinotan
- Roksindol
- RU-24969
- S-14506
- S-14671
- S-15535
- Sarizotan
- Serotonin (5-HT)
- SSR-181507
- Sunepitron
- Triptamini (npr., 5-CT, 5-MeO-DMT, 5-MT, bufotenin, DMT, indorenat, N-Me-5-HT, psilocin, psilocibin)
- TGBA01AD
- U-92016-A
- Urapidil
- Vilazodon
- Ksaliproden
- Johimbin
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- Pozitivni alosterni modulatori: Oleamid
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- Antagonisti: Atipični antipsihotici (npr. iloperidon, risperidon, sertindol)
- AV965
- Beta blokatori (npr. alprenolol, karteolol, cijanopindolol, jodocijanopindolol, isamoltan, oksprenolol, penbutolol, pindobind, pindolol, propranolol, tertatolol)
- BMY-7378
- CSP-2503
- Dotarizin
- Ergolini (npr., metergolin)
- FCE-24379
- Flopropion
- GR-46611
- Isamoltan
- Lekozotan
- Mefway
- Metitepin (metiotepin)
- MIN-117 (WF-516)
- MPPF
- NAN-190
- Robalzotan
- S-15535
- SB-649915
- SDZ 216-525
- Spiperon
- Spiramid
- Spiroksatrin
- UH-301
- WAY-100135
- WAY-100635
- Ksilamidin
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- Agonisti: Anpirtolin
- CGS-12066A
- CP-93129
- CP-94253
- CP-122288
- CP-135807
- Eltoprazin
- Ergolini (npr. bromokriptin, dihidroergotamin, ergotamin, metilergometrin (metilergonovin), metisergid, pergolid)
- mCPP
- RU-24969
- Serotonin (5-HT)
- Triptan (npr. avitriptan, donitriptan, eletriptan, sumatriptan, zolmitriptan)
- TFMPP
- Triptamini (npr. 5-BT, 5-CT, 5-MT, DMT)
- Vortioksetin
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5-HT2 | |
- Agonisti : Serija 25H/NB (npr. 25I-NBF, 25I-NBMD, 25I-NBOH, 25I-NBOMe, 25B-NBOMe, 25C-NBOMe, 25TFM-NBOMe, 2CBCB-NBOMe, 25CN-NBOH, 2CBFly-NBOMe)
- 2C (npr. 2C-B, 2C-E, 2C-I, 2C-T-2, 2C-T-7, 2C-T-21)
- 2C-B-FLY
- 2CB-Ind
- 5-Metoksitriptamini (5-MeO-DET, 5-MeO-DiPT, 5-MeO-DMT, 5-MeO-DPT, 5-5-Metoksitriptamin)
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- Antagonisti: 5-I-R91150
- 5-MeO-NBpBrT
- AC-90179
- Adatanserin
- Altanserin
- Antihistaminici (npr. ciproheptadin, hidroksizin, ketotifen, perlapin)
- AMDA
- Atipični antipsihotici (npr. amperozid, aripiprazol, asenapin, blonanserin, brekspiprazol, karpipramin, klokapramin, klorotepin, klozapin, fluperlapin, gevotrolin, iloperidon, lurasidon, melperon, mosapramin, okaperidon, olanzapin, paliperidon, kvetiapin, risperidon, sertindol, zikronapin, ziprasidon, zotepin)
- Hlorprotiksen
- Cinanserin
- CSP-2503
- Deramciklan
- Dotarizin
- Eplivanserin
- Ergolini (npr. amesergid, LY-53857, LY-215840, mesulergin, metergolin, metisergid, sergoleksol)
- Fananserin
- Flibanserin
- Glemanserin
- Irindalon
- Ketanserin
- KML-010
- Landipirdin
- LY-393558
- mCPP
- Medifoksamin
- Metitepin (metiotepin)
- MIN-117 (WF-516)
- Naftidrofuril
- Nantenin
- Nelotanserin
- Opiranserin (VVZ-149)
- Pelanserin
- Fenoksibenzamin
- Pimavanserin
- Pirenperon
- Pizotifen
- Pruvanserin
- Rauwolscin
- Ritanserin
- Roluperidon
- S-14671
- Sarpogrelat
- Antagonisti serotonina i inhibitori ponovnog preuzimanja (npr. etoperidon, hidroksinefazodon, lubazodon, mepiprazol, nefazodon, triazoledion, trazodon)* SR-46349B
- TGBA01AD
- Teniloksazin
- Temanogrel
- Tetraciklički antidepresivi (npr. amoksapin, aptazapin, esmirtazapin, maprotilin, mianserin, mirtazapin)
- Triciklički antidepresivi (npr. amitriptilin)
- Tipični antipsihotici (npr. hlorpromazin, flufenazin, haloperidol, loksapin, perfenazin, pimozid, pipamperon, prohlorperazin, setoperon, spiperon, spiramid, tioridazin, tiotiksen, trifluoperazin)
- Volinanserin
- Ksilamidin
- Johimbin
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- Agonisti: 4-Metilaminoreks
- Aminoreks
- Amfetamini (npr., klorfentermin, kloforeks, deksfenfluramin, fenfluramin, levofenfluramin, norfenfluramin)
- BW-723C86
- DOx (npr., DOB, DOC, DOI, DOM)
- Ergolin (npr., kabergolin, dihidroergokriptin, dihidroergotamin, ergotamin, metilergometrin (metilergonovin), metisergid, pergolid)
- Lorkaserin
- MDxx (npr., MDA (tenamfetamin), MDMA (midomafetamin), MDOH, MMDA)
- Piperazins (npr., TFMPP)
- PNU-22394
- Ro60-0175
- Serotonin (5-HT)
- Triptamini (npr., 5-BT, 5-CT, 5-MT, α-Me-5-HT, bufotenin, DET, DiPT, DMT, DPT, psilocin, psilocibin, triptamin)
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- Antagonisti: Agomelatin
- Atipični antipsihotici (npr. amisulprid, aripiprazol, asenapin, brekspiprazol, kariprazin, klozapin, N-desalkilkvetiapin (norkvetiapin), N-desmetilklozapin (norklozapin), olanzapin, pipamperon, kvetiapin, risperidon, ziprasidon)
- Ciproheptadin
- EGIS-7625
- Ergolini (npr. amesergid, bromokriptin, lisurid, LY-53857, LY-272015, mesulergin)
- Ketanserin
- LY-393558
- mCPP
- Metadoksin
- Metitepin (metiotepin)
- Pirenperon
- Pizotifen
- Propranolol
- PRX-08066
- Rauwolscin
- Ritanserin
- RS-127445
- Sarpogrelat
- SB-200646
- SB-204741
- SB-206553
- SB-215505
- SB-221284
- SB-228357
- SDZ SER-082
- Tegaserod
- Tetraciklički antidepresivi (npr. amoksapin, mianserin, mirtazapin)
- Trazodon
- Tipični antipsihotici (npr. hlorpromazin)
- TIK-301
- Johimbin
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- Agonisti: 2C (npr., 2C-B, 2C-E, 2C-I, 2C-T-2, 2C-T-7, 2C-T-21)
- 5-Metoksitriptamin (5-MeO-DET, 5-MeO-DiPT, 5-MeO-DMT, 5-MeO-DPT, 5-MT)
- α-alkiltriptamin (npr., 5-Cl-αMT, 5-Fl-αMT, 5-MeO-αET, 5-MeO-αMT, α-Me-5-HT, αET, αMT)
- A-372159
- AL-38022A
- Alstonin
- CP-809101
- Dimemebfe
- DOx (npr. DOB, DOC, DOI, DOM)
- Ergolin (npr. ALD-52, kabergolin, dihidroergotamin, ergin (LSA), ergotamin, lisurid, LA-SS-Az, LSB, LSD, LSD-Pip, LSH, LSP, pergolid)
- Flumeksadol
- Lorkaserin
- MDxx (npr. MDA (tenamfetamin), MDMA (midomafetamin), MDOH, MMDA)
- MK-212
- ORG-12962
- ORG-37684
- Oksaflozan
- PHA-57378
- Fenetilamini (npr. lofofin, meskalin)
- Piperazin (npr. aripiprazol, BZP, mCPP, kvipazin, TFMPP)
- PNU-22394
- PNU-181731
- Ro60-0175
- Ro60-0213
- Serotonin (5-HT)
- Triptamini (npr., 5-BT, 5-CT, bufotenin, DET, DiPT, DMT, DPT, psilocin, psilocibin, triptamin)
- Vabicaserin
- WAY-629
- WAY-161503
- YM-348
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- Antagonisti: Adatanserin
- Agomelatin
- Atipični antipsihotici (npr. asenapin, klorotepin, klozapin, fluperlapin, iloperidon, melperon, olanzapin, paliperidon, kvetiapin, risperidon, sertindol, ziprasidon, zotepin)
- Kaptodiam
- CEPC
- Cinanserin
- Ciproheptadin
- Deramciklan
- Desmetramadol
- Dotarizin
- Eltoprazin
- Ergolin (npr. amesergid, bromokriptin, LY-53857, LY-215840, mesulergin, metergolin, metisergid, sergoleksol)
- Etoperidon
- Fluoksetin
- FR-260010
- Irindalon
- ketanserin
- ketotifen
- Latrepirdin (dimebolin)
- Medifoksamin
- Metitepin (metiotepin)
- Nefazodone
- Pirenperone
- Pizotifen
- Propranolol
- Ritanserin
- RS-102221
- S-14671
- SB-200646
- SB-206553
- SB-221284
- SB-228357
- SB-242084
- SB-243213
- SDZ SER-082
- Tedatioksetin
- Tetraciklički antidepresivi (npr. amoksapin, aptazapin, esmirtazapin, maprotilin, mianserin, mirtazapin)
- TIK-301
- Tramadol
- Trazodon
- Triciklički antidepresivi (npr. amitriptilin, nortriptilin)
- Tipični antipsihotici (npr. klorpromazin, loksapin, pimozid, pipamperon, tioridazin)
- Ksilamidin
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5-HT3–7 | | |
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- Agonisti : Ergolini (npr. dihidroergokriptin, dihidroergotamin, ergotamin, lisurid, LSD, mesulergin, metergolin, metisergid)
- Hipidon
- Serotonin (5-HT)
- Triptamini (npr. 2-Me-5-HT, 5-BT, 5-CT, 5-MT, bufotenin, E-6801, E-6837, EMD-386088, EMDT, LY-586713, N-Me-5-HT, ST-1936, triptamin)
- WAY-181187
- WAY-208466
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- Negativni alosterni modulatori: Oleamid
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